Tohoku J. Exp. Med., 2000, 191 (3)

Induction of Tissue Factor Production but not the Upregulation of Adhesion Molecule Expression by Ceramide in Human Vascular Endothelial Cells

MAKOTO HIROKAWA, ATSUSHI KITABAYASHI, JUN KUROKI and AKIRA B. MIURA

The Third Department of Internal Medicine, Akita University School of Medicine, Akita 010-8543

  • Binding of tumor necrosis factor-a (TNF-a) to p60 TNF-a receptor induces the activation of sphingomyelinase to generate ceramide, which in turn activates certain protein kinases and phosphatases, resulting in various TNF-a-mediated biological effects. We have investigated the role for the sphingomyelin/ceramide pathway in the TNF-a-induced upregulation of adhesion molecule expression and tissue factor production of human endothelial cells. TNF-a stimulated human umbilical vascular endothelial cells (HUVECs) to upregulate the expression of vascular cell adhesion molecule-1 (VCAM-1), intercellular adhesion molecule-1 (ICAM-1) and HLA class I molecules in addition to the induction of procoagulant tissue factor production. C2-ceramide, a highly cell-permeable ceramide analog, was able to stimulate HUVECs to produce tissue factor activity as well as TNF-a. However, C2-ceramide did not stimulate HUVECs to upregulate the expression of VCAM-1, ICAM-1 and HLA class I molecules. These results suggest that there exist both the ceramide-dependent and -independent pathways in TNF-a signal transduction system in human vascular endothelial cells.
    Key words--- human endothelial cells; TNF-a; ceramide; tissue factor; adhesion molecules
    © 2000 Tohoku University Medical Press


    Tohoku J. Exp. Med., 2000, 191, 167-176
    Address for reprints: Makoto Hirokawa, M.D., Division of Hematology, The Third Department of Internal Medicine, Akita University School of Medicine, 1-1-1 Hondo, Akita 010-8543, Japan.
    e-mail: hirokawa@med.akita-u.ac.jp


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